ChloroquineV1, France, Analysis, bibRecord, 000218

Ugi-Smiles couplings of 4-substituted pyridine derivatives: A fast access to chloroquine analogues

Identifieur interne : 000218 ( France/Analysis ); précédent : 000217; suivant : 000219

Ugi-Smiles couplings of 4-substituted pyridine derivatives: A fast access to chloroquine analogues

Auteurs : Laurent El Kaim [France] ; Laurence Grimaud [France] ; Patil Pravin [France]

Source :

Organic Letters [ 1523-7060 ] ; 2012.

RBID : Hal:hal-00949992

Abstract

4-Hydroxy and mercapto pyridines were successfully tested in Ugi-Smiles couplings. Such multicomponent reactions applied to quinoline derivatives afford a very convenient and short synthesis of antimalarial analogues. © 2011 American Chemical Society.

Url:

https://hal-polytechnique.archives-ouvertes.fr/hal-00949992

DOI: 10.1021/ol202974w

Affiliations:

France

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to stream Hal, to step Corpus: 000247
to stream Hal, to step Curation: 000247
to stream Hal, to step Checkpoint: 000157
to stream Main, to step Merge: 001287
to stream Main, to step Curation: 001286
to stream Main, to step Exploration: 001286
to stream France, to step Extraction: 000218

Links to Exploration step

Hal:hal-00949992

Le document en format XML

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   |texte=   Ugi-Smiles couplings of 4-substituted pyridine derivatives: A fast access to chloroquine analogues
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Ugi-Smiles couplings of 4-substituted pyridine derivatives: A fast access to chloroquine analogues

Ugi-Smiles couplings of 4-substituted pyridine derivatives: A fast access to chloroquine analogues

Source :

Abstract

Links toward previous steps (curation, corpus...)

Links to Exploration step

Le document en format XML

Pour manipuler ce document sous Unix (Dilib)

Pour mettre un lien sur cette page dans le réseau Wicri